Grazioso Giovanni
Associate Professor
Scientific-Disciplinary Sector
CHEM-07/A - Pharmaceutical Chemistry
Scientific-Disciplinary Group/Competition Sector
03/CHEM-07 - CHIMICA FARMACEUTICA, TOSSICOLOGICA, NUTRACEUTICO-ALIMENTARE, DELLE FERMENTAZIONI E DEI PRODOTTI PER IL BENESSERE E PER LA SALUTE
Research fields and competencies
Contacts
Workplace
Office phone number
Additional phone numbers
University email address
Office hours
every day by prior arrangement made via email
Reception office
Office 2015 - Lab. 2053 - Via L. Mangiagalli 25
Teaching - Programme courses
Bachelors and masters
A.Y. 2025/2026
A.Y. 2024/2025
A.Y. 2023/2024
A.Y. 2022/2023
A.Y. 2021/2022
A.Y. 2020/2021
Postgraduate programmes
A.Y. 2024/2025
Doctoral programme (PhD)
A.Y. 2023/2024
Doctoral programme (PhD)
A.Y. 2022/2023
Doctoral programme (PhD)
Research
Publications
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Enhancing the activity of γ-hydroxy lactone derivatives as innovative peroxisome proliferator-activated receptor γ non-agonists inhibiting cyclin-dependent kinase 5-mediated phosphorylation / G. Cazzaniga, D. Capelli, R. Montanari, E.M.A. Fassi, G. Grazioso, A. Tresoldi, F. Rinaldi, E. Calleri, I. Bassanini, S. Romeo, M. Garofalo, M. Mori, F. Meneghetti, S. Villa. - In: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. - ISSN 0223-5234. - 292:(2025 Aug 05), pp. 117657.1-117657.18. [10.1016/j.ejmech.2025.117657]
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FYCO1 Peptide Analogs: Design and Characterization of Autophagy Inhibitors as Co-Adjuvants in Taxane Chemotherapy of Prostate Cancer / E.M.A. Fassi, R.M. Moretti, M. Montagnani Marelli, M. Garofalo, A. Gori, C. Pesce, M. Albani, E.G. Milano, J. Sgrignani, A. Cavalli, G. Grazioso. - In: INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES. - ISSN 1422-0067. - 26:11(2025 Jun 03), pp. 5365.1-5365.22. [10.3390/ijms26115365]
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Insights on Zosteric Acid Analogues Activity Against Candida albicans Biofilm Formation / C. Catto', E.M.A. Fassi, G. Grazioso, A. Gelain, S. Villa, F. Cappitelli. - In: ACS OMEGA. - ISSN 2470-1343. - 10:21(2025 May 20), pp. 22285-22295. [10.1021/acsomega.5c03581]
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A potent nonapeptide inhibitor for the CXCL12/HMGB1 heterocomplex: A computational and experimental approach / E.M.A. Fassi, E. Pirani, V. Cecchinato, A. Cavalli, G. Roda, M. Uguccioni, J. Sgrignani, G. Grazioso. - In: COMPUTATIONAL AND STRUCTURAL BIOTECHNOLOGY JOURNAL. - ISSN 2001-0370. - 27:(2025 Apr 25), pp. 1677-1685. [10.1016/j.csbj.2025.04.023]
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Exploiting the Potential of Computational Approaches in Medicinal Chemistry: CADD of Novel eIF6 Binders for the Development of anti-HCC PROTACs / A. Colleoni, E.M.A. Fassi, A. Miluzio, G. Tempra, M. Albani, M. DE AMICI, G. Grazioso, S. Biffo, C. Matera. ((Intervento presentato al convegno WIDEnzymes : 27th – 31st January tenutosi a Lecco nel 2025.