Taramelli Donatella

Novel antimalarial 3-substituted quinolones isosteres with improved pharmacokinetic properties / S. Ge, R. Jian, Q. Xuan, Y. Zhu, X. Ren, W. Li, X. Chen, R.K. Huang, C.S. Lee, S.C. Leung, N. Basilico, S. Parapini, D. Taramelli, N. Pinthong, S.V. Antonyuk, P.M. O'Neill, Z. Sheng, W.D. Hong. - In: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. - ISSN 0223-5234. - 284:(2025 Feb 15), pp. 117228.1-117228.12. [10.1016/j.ejmech.2024.117228]

Design, synthesis and modelling of photoreactive chemical probes for investigating target engagement of plasmepsin IX and X in Plasmodium falciparum / M. Lisauskaitė, G.L. Nixon, C.M. Woodley, N.G. Berry, A. Coninckx, L. Charlie Qie, S.C. Leung, D. Taramelli, N. Basilico, S. Parapini, S.A. Ward, O. Vadas, D. Soldati-Favre, W. David Hong, P.M. O'Neill. - In: RSC CHEMICAL BIOLOGY. - ISSN 2633-0679. - 5:1(2024), pp. 19-29. [10.1039/D3CB00109A]

Favorable Preclinical Pharmacological Profile of a Novel Antimalarial Pyrrolizidinylmethyl Derivative of 4-amino-7-chloroquinoline with Potent In Vitro and In Vivo Activities / N. Basilico, S. Parapini, S. D’Alessandro, P. Misiano, S. Romeo, G. Dondio, V. Yardley, L. Vivas, S. Nasser, L. Rénia, B.M. Russell, R. Suwanarusk, F. Nosten, A. Sparatore, D. Taramelli. - In: BIOMOLECULES. - ISSN 2218-273X. - 13:5(2023 May 14), pp. 836.1-836.23. [10.3390/biom13050836]

In-vitro antiviral activity and in-silico targeted study of quinoline-3-carboxylate derivatives against SARS-Cov-2 isolate / R.K. Mittal, P. Purohit, M. Sankaranarayanan, M. Muzaffar-Ur-Rehman, D. Taramelli, L. Signorini, M. Dolci, N. Basilico. - In: MOLECULAR DIVERSITY. - ISSN 1381-1991. - (2023), pp. 1-15. [Epub ahead of print] [10.1007/s11030-023-10703-w]

From DC18 to MR07: A Metabolically Stable 4,4′‐Oxybisbenzoyl Amide as a Low‐Nanomolar Growth Inhibitor of P. falciparum / I. Bassanini, S. Parapini, N. Basilico, D. Taramelli, S. Romeo. - In: CHEMMEDCHEM. - ISSN 1860-7179. - 17:21(2022 Nov 04), pp. 1-9. [10.1002/cmdc.202200355]